产品编号 | 产品名称 | CAS No. |
DC8648 |
Rev-erbα agonist GS4112
GSK4112 is a Rev-erbα agonist with EC50 of 0.4 μM, also is a small molecule chemical probe for the cell biology of the nuclear heme receptor Rev-erbα. |
1216744-19-2 |
DC8649 |
1-Methyl-7-nitroisatoic anhydride
1-methyl-7-nitroisatoic anhydride is a reagent that detects local nucleotide flexibility, for probing 2'-hydroxyl reactivity. |
73043-80-8 |
DC8693 |
Epiandrosterone
Epiandrosterone is a steroid hormone with weak androgenic activity. Epiandrosterone is naturally produced by the enzyme 5α-reductase from the adrenal hormone DHEA. |
481-29-8 |
DC8701 |
Fmoc-Val-Cit-PAB-PNP
Fmoc-Val-Cit-PAB-PNP is a peptide prodrug linker, is a linker for antibody-drug-conjugation (ADC). |
863971-53-3 |
DC8710 |
Tranylcypromine HCl
Tranylcypromine HCl is an inhibitor of monoamine oxidase (MAO) and prostacyclin synthase, potently suppresses the enzymatic activity of Lysine-Specific Demethylase 1 (LSD1) (IC50 <2 μM for BHC110/LSD1). |
1986-47-6 |
DC8735 |
AHU-377 hemicalcium salt
AHU-377 is an inhibitor of neprilysin with IC50 value of 5 nM. |
1369773-39-6 |
DC8737 |
SCH900776 S-isomer
SCH900776 (S-isomer) is the S-isomer form of SCH900776, which is a potent, selective and orally bioavailable inhibitor of checkpoint kinase Chk1 (IC50 = 3 nM), highly selective against Chk2 (IC50 = 1500 nM) and cyclin-dependent kinase CDK2 (IC50 |
891494-64-7 |
DC8738 |
Sal003
Sal003 is a potent cell-permeable analog of the eIF2α phosphatase inhibitor Salubrinal with enhanced aqueous solubility. |
1164470-53-4 |
DC8747 |
PD-151746
PD 151746 is a selective, cell-permeable calpain inhibitor with Ki of 0.26 μM for μ-Calpain, about 20-fold selectivity over m-calpain. |
179461-52-0 |
DC8755 | WAY 100635 Hydrochloride | 146714-97-8 |
DC8766 |
GSK1324726A (I-BET726)
GSK1324726A In stock,price: 680 USD/100mg. GSK1324726A (I-BET726) is a novel, potent, and selective small molecule inhibitor of BET proteins with high affinity to BRD2 (IC50= 41 nM), BRD3 (IC50= 31 nM), and BRD4 (IC50= 22 nM). |
1300031-52-0 |
DC8779 |
Glycopyrrolate
Glycopyrrolate(Glycopyrronium Br) is a muscarinic competitive antagonist used as an antispasmodic. |
596-51-0 |
DC8791 |
Sorafenib free base (BAY-43-9006)
Sorafenib(BAY 43-9006) is a potent inhibitor of Raf-1 with IC50 values of 6 nM, 22 nM and 90 nM for Raf-1, B-Raf, and VEGFR2 respectively, BAY 43-9006 suppresses both wild-type and V599E mutant BRAF activity in vitro. |
284461-73-0 |
DC8792 |
Pirfenidone(AMR69)
Pirfenidone(AMR69) is an inhibitor for TGF-β production and TGF-β stimulated collagen production, reduces production of TNF-α and IL-1β, and also has anti-fibrotic and anti-inflammatory properties. Phase 3. |
53179-13-8 |
DC8855 |
Fumagillin
Fumagillin is a selective and potent irreversible inhibitor of Methionine aminopeptidase 2 (MetAP2), used as an antibiotic to treat microsporidiosis. |
23110-15-8 |
DC8856 |
EPI-001
EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ∼6 μM and a selective PPAR-gamma modulator |
227947-06-0 |
DC8876 |
Rimonabant(SR141716)
Rimonabant(SR141716) is a selective central cannabinoid (CB1) receptor inverse agonist with Ki of 1.8 nM. |
168273-06-1 |
DC8895 |
benzbromaron
Benzbromarone is a highly effective and well tolerated non-competitive inhibitor of xanthine oxidase, used as an uricosuric agent, used in the treatment of gout. |
3562-84-3 |
DC8900 |
SRT1720
SRT1720 is a selective activator of human SIRT1 (EC1.5 = 0.16 μM) versus the closest sirtuin homologues, SIRT2 and SIRT3 (SIRT2: EC1.5 = 37 μM;SIRT3: EC1.5 > 300 μM). |
925434-55-5 |
DC8925 |
Atipamezole
Atipamezole(MPV1248) is an alpha-adrenoceptor antagonist with high affinity and selectivity for the alpha 2-receptor. |
104054-27-5 |
DC8928 |
Minocycline hydrochloride
Minocycline is a tetracycline antibiotic with neuroprotective, antiapoptotic, anti-inflammatory and antimicrobial effects. |
13614-98-7 |
DC8935 |
Mitomycin C
Mitomycin C is a DNA crosslinking agent that inhibits DNA synthesis and induces apoptosis in a variety of cells. |
1950-7-7 |