产品编号 | 产品名称 | CAS No. |
DC10573 |
MDK34597 (PI3K inhibitor)
Featured
MDK34597 is a PI3K inhibitor.MDK34597 is an analog of PI-103 and acts as a dual PI3K/mTOR Inhibitor. |
371934-59-7 |
DC10574 |
CID-25014542
Featured
5-chloro-3-(3,5-dibromo-4-hydroxybenzylidene)indolin-2-one |
220904-99-4 |
DC10575 |
Methyl 13-cis-4-Oxoretinoate
Featured
methyl (2Z,4E,6E,8E)-3,7-dimethyl-9-(2,6,6-trimethyl-3-oxocyclohexen-1-yl)nona-2,4,6,8-tetraenoate |
71748-57-7 |
DC10576 |
Cyantraniliprole
Featured
Cyantraniliprole(HGW-86)是一具杀昆虫剂性质化合物。 |
736994-63-1 |
DC10577 |
ADT-OH
Featured
ADT-OH是茴香脑二硫代硫酮(ADT)和合成硫化氢(H2S)供体的衍生物。 在体外葡萄糖 - 氧剥夺(OGD)模型中,ADT-OH显着减弱tPA增强的Akt活化和脑微血管内皮细胞中的VEGF表达。 最后,ADT-OH改善了MCAO和tPA输注小鼠的功能结果。 H2S供体通过可能抑制Akt-VEGF-MMP9级联来减少tPA诱导的脑出血。 施用H2S供体具有作为改善中风后tPA安全性的新方式的潜力。 |
18274-81-2 |
DC10578 |
rac BHFF
Featured
Rac BHFF is a potent and selective GABAB receptor positive allosteric modulator that increases the efficacy and potency of GABA ( > 149% and > 15-fold respectively). Orally active and exhibits anxiolytic activity in vivo. |
123557-91-5 |
DC10579 |
CAY 10602
Featured
CAY10602 是一个 SIRT1 激活剂。 |
374922-43-7 |
DC1058 |
LY294002
Featured
LY294002 (NSC 697286; SF 1101) 是一种广谱 PI3K 抑制剂,抑制 PI3Kα, PI3Kδ 和 PI3Kβ 的 IC50 分别为 0.5, 0.57, 0.97 μM。LY294002 也可抑制 CK2 的活性,IC50 为 98 nM。LY294002 是一种竞争性 DNA-PK 抑制剂,可逆结合 DNA-PK 的激酶结构域,IC50 为 1.4 μM。LY294002 是一种自噬 (autophagy) 和凋亡 (apoptosis) 激活剂。 |
154447-36-6 |
DC10580 |
hVEGF-IN-1
Featured
hVEGF-IN-1抑制人类 VEGF-A 翻译,具有抗肿瘤活性。 |
1637443-98-1 |
DC10581 |
Succinobucol(AGI 1067)
Featured
Succinobucol 是一种酚类抗氧化剂,具有抗炎、抗血小板聚集的作用。 |
216167-82-7 |
DC10582 |
Diroximel Fumarete(ALKS-8700)
Featured
Diroximel fumarate (DRF) 是富马酸单乙酯 (MMF) 的前体药物,是一种控释制剂,可在体内迅速有效的转化为 MMF。 |
1577222-14-0 |
DC10583 |
RO 5028442
Featured
RG7713 (RO5028442) 是一种高效且有选择性的脑-渗透加压素 1a (V1a) 受体拮抗剂,其 Ki 值为 1 nM (hV1a) 和 39 nM (mV1a)。 |
920022-47-5 |
DC10584 |
IRAK4-IN-1
Featured
IRAK4-IN-1 是白细胞介素-1 受体相关激酶 4 (IRAK4) 抑制剂,IC50 为 7 nM。 |
1820787-94-7 |
DC10585 |
Hispidol
Featured
Hispidol ((Z)-Hispidol) 是炎症性肠病的潜在治疗剂;抑制 TNF-α 诱导的单核细胞对结肠上皮细胞的粘附,IC50 值为0.50 µM。 |
5786-54-9 |
DC10586 |
KDM4D-IN-1
Featured
KDM4D-IN-1 是一种新型组蛋白赖氨酸去甲基化酶 4D (KDM4D) 抑制剂,IC50 为 0.41±0.03 μM。 |
2098902-68-0 |
DC10587 |
SPI 112
Featured
SPI 112 is novel Shp2 PTP inhibitor. |
1051387-90-6 |
DC10588 |
ASP-9521
Featured
ASP-9521是有效,选择性,有口服活性的AKR1C3抑制剂;对人类AKR1C3的IC50值为11 nM。 |
1126084-37-4 |
DC10589 |
AG 1406
Featured
AG 1406 is a selective inhibitor of the receptor tyrosine kinase VEGF receptor 2 . |
71308-34-4 |
DC1059 |
Lumacaftor(vx-809,vx809)
Featured
Lumacaftor (VX-809; VRT 826809) 是 CFTR 调节剂,可纠正 CFTR 蛋白的折叠和运输。 |
936727-05-8 |
DC10590 |
Gemcitabine monophosphate
Featured
Gemcitabine monophosphate |
1638288-31-9 |
DC10591 |
CPI-613
Featured
Devimistat (CPI-613) 是一种硫辛酸类似物,可抑制丙酮酸脱氢酶 (PDH) 和 α-酮戊二酸脱氢酶,破坏线粒体代谢 并显示出强大的抗肿瘤活性。 |
95809-78-2 |
DC10592 |
ASL 601(Acecainide)
Featured
Acecainide, also known as N-acetylprocainamide and ASL 601, is the N-acetylated metabolite of procainamide. |
34118-92-8 |