产品编号 | 产品名称 | CAS No. |
DC10546 |
GNE-495
Featured
GNE-495 是有效,选择性的 MAP4K4 抑制剂,IC50 值3.7 nM。 |
1449277-10-4 |
DC10547 |
Ensartinib
Featured
X-376 是一种有效的高特异性 ALK 酪氨酸激酶抑制剂 (TKI) (IC50=0.61 nM)。X-376 是 MET 的较低效抑制剂 (IC50=0.69 nM)。X-376 具有有效的抗肿瘤活性。 |
1365267-27-1 |
DC10548 |
Auten-99
Featured
Auten-99 is a novel inhibitor of the myotubularin phosphatase Jumpy (also called MTMR14), acrossing the blood-brain barrier and exerting potent neuroprotective effects. |
1049780-58-6 |
DC10549 |
Nomifensine maleate
Featured
Nomifensine maleate是多巴胺摄取的选择性抑制剂,治疗成人注意力缺陷障碍。 |
32795-47-4 |
DC10550 |
DKM 2-93
Featured
DKM 2-93是相对选择性的UBA5抑制剂,IC50值为430 μM。 |
65836-72-8 |
DC10551 |
Necrostatin 2 racemate
Featured
Necrostatin 2 racemate (Nec-1S),是一种稳定型 Nec-1 (HY-15760 ),Necrostatin 2 racemate 是一种有效且特异性的 RIPK1 抑制剂,但缺乏 IDO 靶向作用。 |
852391-15-2 |
DC10552 |
AU1235
Featured
AU1235是结核分枝杆菌金刚烷脲尿素抑制剂。 |
1338780-86-1 |
DC10553 |
ST034307
Featured
ST034307 是一种有效的,选择性的 adenylyl cyclase 1 抑制剂,IC50 值为 2.3 μM。 |
133406-29-8 |
DC10554 |
DC260126
Featured
DC260126 是一种 GPR40 拮抗剂。 |
346692-04-4 |
DC10555 |
inS3-54A18
Featured
inS3-54A18 是有一种有效的 STAT3 抑制剂,具有抗癌作用。 |
328998-53-4 |
DC10556 |
KY1220
Featured
KY1220作用于 Wnt/β-catenin 靶点,使β-catenin 和 Ras不稳定。在HEK293报告细胞中的IC50 值为2.1 μM。 |
292168-79-7 |
DC10557 |
ML402
Featured
ML402 是选择性的 TREK-1 激活剂。 |
298684-44-3 |
DC10558 |
ASP 7663
Featured
(2E)-(7-Fluoro-1-isobutyl-2-oxo-1,2-dihydro-3H-indol-3-ylidene)acetic acid |
1190217-35-6 |
DC1056 |
PD0325901 (PD325901)
Featured
PD0325901是选择性,可渗透细胞的 MEK 抑制剂, IC50为0.33 nM。 |
391210-10-9 |
DC10560 |
MAK683
Featured
MAK683 是胚胎外胚层发育 (EED) 抑制剂,来自专利US20160176882 A1,化合物实例 2;在EED Alphascreen,LC-MS 和 ELISA 试验中的 IC50 值分别为 59,89,26 nM。 |
1951408-58-4 |
DC10567 |
KKL-10
Featured
KKL-10是一种具有广谱抗菌活性的小分子核糖体拯救抑制剂。 |
952849-76-2 |
DC10568 |
Mitapivat
Featured
Mitapivat 是一种丙酮酸激酶 M2 型同工酶 (PKM2) 激活剂。 |
1260075-17-9 |
DC10569 |
MDK1088(T.cruzi Inhibitor)
Featured
MDK-1088, also known as T.cruzi Inhibitor, is a Trypanosoma cruzi inhibitor. MDK-1088 has CAS#1350920-22-7 . The last 4 digit f CAS# was used in its name. |
1350920-22-7 |
DC1057 |
Fidaxomicin (Dificid)
Featured
Fidaxomicin (OPT-80) 是一种大环 RNA 聚合酶抑制剂,具有窄谱活性。 Fidaxomicin 选择性地根除致病性艰难梭菌 (Clostridium difficile),对构成正常健康肠道菌群的多种细菌的破坏程度最小。 |
873857-62-6 |
DC10570 |
MDK74978(Multi-kinase inhibitor)
Featured
N-(2-Hydroxyethyl)-4-(6-{[4-(trifluoromethoxy)phenyl]amino}-4-pyrimidinyl)benzamide |
778274-97-8 |
DC10571 |
MDK-8582(Hnps-PLA Inhibitor)
Featured
MDK-8582, also known as Hnps-PLA Inhibitor, is an nhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA). |
185298-58-2 |
DC10572 |
MDK35833(Oct3/4-inducer-1)
Featured
{4-[(4-Fluorobenzyl)oxy]phenyl}acetonitrile |
1016535-83-3 |