产品编号 | 产品名称 | CAS No. |
DC12145 |
DLinDMA
Featured
DLinDMA is a key lipid component of stable nucleic acid lipid particles as a benchmark. |
871258-12-7 |
DC12191 |
JQ-35-(S)
Featured
JQ-35, (S)- is an inhibitor of the Bromodomain and Extra-Terminal (BET) family bromodomain-containing proteins with potential antineoplastic activity. |
1349719-98-7 |
DC12522 |
MKK7-COV-3
Featured
MKK7-COV-3 (MKK7 Covalen inhibitor 3) is a potent, selective, covalent MKK7 inhibitor with in vitro IC50 of 5 nM, displays >1,000-fold selectivity over MKK4 (IC50=7.81 uM). |
|
DC12526 |
OGG1 inhibitor O8
Featured
OGG1 inhibitor O8 is a potent, selective inhibitor of 8-oxoguanine DNA glycosylase 1 (OGG1) with IC50 of 0.22 uM, |
350997-39-6 |
DC12541 |
iGOT1-01
Featured
iGOT1-01 is a small molecule inhibitor of aspartate aminotransferase 1 (glutamate oxaloacetate transaminase 1 (GOT1)) with IC50 of 11.3 uM. |
882256-55-5 |
DC12542 |
GOT1 inhibitor 2c
Featured
GOT1抑制剂2c是谷氨酸草酰乙酸转氨酶1(GOT1)的一流的非共价抑制剂,IC50为8.2μM。 |
732973-87-4 |
DC12568 |
UBCS039
Featured
UBCS039 (UBCS-039) is the first synthetic activator of the NAD+-dependent protein lysine deacetylase SIRT6 with EC50 of 38 uM. |
358721-70-7 |
DC20000 |
LR-90
Featured
LR-90 is an advanced glycation end product (AGE) inhibitor, inhibits inflammatory responses in human monocytes. LR-90 is also used in the research of diabetic animal model. |
245075-84-7 |
DC20332 |
CD38 inhibitor 78c
Featured
CD38 inhibitor 78c is a potent, specific, reversible CD38 inhibitor with Ki of 14.5 nM for recombinant human CD38. |
1700637-55-3 |
DC20446 |
Mefuparib hydrochloride
Featured
Mefuparib hydrochloride is a potent, highly selective, competitive PARP1/2 inhibitor with IC50 of 3.2/1.9 nM, respectively. |
1449746-00-2 |
DC20613 |
A-800141
Featured
A-800141 is a potent, highly specific, orally bioavailable MetAP2 inhibitor with IC50 of 12 nM, shows no inhibition for MetAP1 (IC50>30 uM). |
681245-85-2 |
DC2107 |
Gemcitabine HCl (Gemzar,LY188011)
Featured
Gemcitabine Hydrochloride (Gemzar) is a DNA synthesis inhibitor ,showed potent activity against COVID-19(SARS-COV-2) with EC50 MERS-COV(1.216), SARS-COV(4.957). |
122111-03-9 |
DC21158 |
JAK3-IN-2
Featured
A potent and highly selective JAK3 inhibitor with IC50 of 0.15 nM. |
1443235-95-7 |
DC21396 |
Marizomib
Featured
A potent, orally bioactive 20S proteasome inhibitor with IC50 of 1.3 nM (inhibition of proteasomal chymotrypsin-like proteolytic activity). |
437742-34-2 |
DC21567 |
Triazavirin
Featured
Triazavirin (Riamilovir sodium dihydrate) is a broad-spectrum antiviral agent targeting influenza viruses, lassa virus, TBEV and Ebola virus. |
928659-17-0 |
DC21593 |
RUC-4
Featured
A potent, selective, non-RGD-mimetic αIIbβ3 integrin receptor antagonist with IC50 of 45 nM, with no activity on αVβ3 receptors. . |
1448313-27-6 |
DC21869 |
Borussertib
Featured
Borussertib is a potent, first-in-class, covalent-allosteric AKT inhibitor. |
1800070-77-2 |
DC22453 |
Sappanone A
Featured
A homoisoflavanone found in Caesalpinia sappan, a potent, selective IMPDH2 inhibitor that covalently binds to Cys140 with Kd of 3.944 nM, almost 10 times lower than the Kd of binding to IMPDH1. |
102067-84-5 |
DC22637 |
BKI1369
Featured
BKI-1369 is an effective bumped kinase inhibitor (BKI), inhibits Theileria equi in vitro and reduces parasite burden and disease severity in the gnotobiotic pig model. |
1951431-22-3 |
DC22819 |
CCG-50014
Featured
CCG-50014 (CCG50014) is a potent, selective, covalent inhibitor of RGS4 with IC50 of 30 nM. |
883050-24-6 |
DC22938 |
ICA-027243
Featured
A novel potent, selective KCNQ2/Q3 (Kv7.2/Kv7.3) potassium channel opener/activator with EC50 of 0.38 uM.. |
325457-89-4 |
DC23119 |
FB23-2(FTO Demethylase inhibitor FB23-2)
Featured
FB23-2 is a potent, selective inhibitor of the mRNA N 6-methyladenosine (m 6A) demethylase FTO, directly bind to FTO, inhibits FTO demethylation of m6 A in RNA in vitro with IC50 of 2.6 uM. |
2243736-45-8 |