Almorexant HCl (Act-078573)
产品编号: DC7692
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应用领域
Almorexant hydrochloride (ACT 078573 hydrochloride) 是一种有效的食欲素受体 orexin 1 receptor (OX1)/orexin 2 receptor (OX2) 拮抗剂,Ki 分别为 1.3 和 0.17 nM。
Cas No.: |
913358-93-7 |
名称: |
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别名: |
ACT-078573; ACT 078573; ACT078573 |
SMILES: |
C(NC)(=O)[C@@H](N1CCC2=C([C@H]1CCC1=CC=C(C(F)(F)F)C=C1)C=C(OC)C(OC)=C2)C1=CC=CC=C1.[H]Cl |
分子式: |
C29H32ClF3N2O3 |
分子量: |
549.02 |
纯度: |
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保存条件: |
2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
Description: |
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References: |
Almorexant(ACT078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.
IC50 value: 1.3/0.7 nM(OX1/OX2 receptor)
Target: Dual OX!/OX2 receptor
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MSDS
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MSDS_1906_DC7692_913358-93-7 |
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