Umeclidinium bromide

产品编号: DC8153 Featured
Umeclidinium bromide
结构式
869113-09-7
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中国地区超过5000个高品质化合物库存
应用领域
Umeclidinium bromide 是一种 mAChR 拮抗剂。Umeclidinium bromide 作用于克隆的人 M1-M5 mAChRs,Ki 为 0.05 到 0.16 nM。
Cas No.: 869113-09-7
名称:
别名:
SMILES: C1C[N+]2(CCC1(CC2)C(C3=CC=CC=C3)(C4=CC=CC=C4)O)CCOCC5=CC=CC=C5.[Br-]
分子式: C29H34BrNO2
分子量: 508.49
纯度:
保存条件: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description:
In Vivo:
In Vitro:
References: Umeclidinium bromide(GSK573719A) is a muscarinic receptor antagonist which is useful in treatment of chronic obstructive pulmonary disease (COPD). For the detailed information of Umeclidinium bromide(GSK573719A), the solubility of Umeclidinium bromide(GSK573719A) in water, the solubility of Umeclidinium bromide(GSK573719A) in DMSO, the solubility of Umeclidinium bromide(GSK573719A) in PBS buffer, the animal experiment (test) of Umeclidinium bromide(GSK573719A), the cell expriment (test) of Umeclidinium bromide(GSK573719A), the in vivo, in vitro and clinical trial test of Umeclidinium bromide(GSK573719A), the EC50, IC50,and affinity,of Umeclidinium bromide(GSK573719A), For the detailed information of Umeclidinium bromide(GSK573719A), the solubility of Umeclidinium bromide(GSK573719A) in water, the solubility of Umeclidinium bromide(GSK573719A) in DMSO, the solubility of Umeclidinium bromide(GSK573719A) in PBS buffer, the animal experiment (test) of Umeclidinium bromide(GSK573719A), the cell expriment (test) of Umeclidinium bromide(GSK573719A), the in vivo, in vitro and clinical trial test of Umeclidinium bromide(GSK573719A), the EC50, IC50,and affinity,of Umeclidinium bromide(GSK573719A), Please contact DC Chemicals.
Kinase Assay:
Cell Assay:
Animal Administration:
References:
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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