Cebranopadol(GRT-6005)
产品编号: DC7097
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应用领域
Cebranopadol 是NOP 和 opioid receptor 激动剂，作用于人NOP，MOP，KOP 和δ-阿片肽(DOP)受体，Ki/EC50 分别为 0.9 nM/13 nM，0.7 nM/1.2 nM，2.6 nM/17 nM，18 nM/110 nM。
| Cas No.: |
863513-91-1 |
| 名称: |
6-fluoro-N,N-dimethyl-1'-phenylspiro[4,9-dihydro-3H-pyrano[3,4-b]indole-1,4'-cyclohexane]-1'-amine |
| 别名: |
GRT-6005; GRT 6005; GRT6005 |
| SMILES: |
CN(C)C1(CCC2(CC1)C3=C(CCO2)C4=C(N3)C=CC(=C4)F)C5=CC=CC=C5 |
| 分子式: |
C24H27FN2O |
| 分子量: |
378.48 |
| 纯度: |
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| 保存条件: |
2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
| Description: |
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| References: |
Cebranopadol has a unique mechanism of action, activating both the NOP (nociceptin/orphanin FQ peptide) receptor and the mu opioid receptor.For the detailed information of Cebranopadol(GRT-6005), the solubility of Cebranopadol(GRT-6005) in water, the solu |
| Kinase Assay: |
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| Cell Assay: |
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| Animal Administration: |
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| References: |
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MSDS
COA
| LOT NO. |
DOWNLOAD |
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| 2018-0101 |
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询盘
