AC-263093

产品编号: DC12577 Featured
AC-263093
结构式
849459-86-5
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中国地区超过5000个高品质化合物库存
应用领域
AC-263093(AC263093)是一种有效的功能选择性神经肽FF受体2型(NPFFR2)激动剂,pKi为6.9;对NPFFR1和NPFFR2显示出相同的亲和力,并且功能性失活的NPFFR1;减弱体内吗啡耐受性。
Cas No.: 849459-86-5
名称: 2-(3,4-dibromobenzylidene)hydrazine-1-carboximidamide
别名: AC263093,AC 263093
SMILES: N(C(N)=N)/N=C/C1=CC=C(Br)C(Br)=C1
分子式: C8H8Br2N4
分子量: 319.988
纯度:
保存条件: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description:
In Vivo:
In Vitro:
References: AC-263093 (AC263093) is a potent, functionally selective neuropeptide FF receptor type 2 (NPFFR2) agonist with pKi of 6.9; shows equal affinity for NPFFR1 and NPFFR2, and functionally inactivated NPFFR1; attenuates morphine tolerance in vivo.
Kinase Assay:
Cell Assay:
Animal Administration:
References:
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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