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Elamipretide (TFA salt)

产品编号: DC21695 Featured
Elamipretide (TFA salt)
结构式
736992-21-5
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中国地区超过5000个高品质化合物库存
应用领域
Elamipretide是一个心磷脂过氧化物酶抑制剂和线粒体靶向的肽，能够提高左心室和线粒体功能。
化学性质生物活性化合物的使用COA & MSDS相关产品产品说明书
Cas No.: 736992-21-5
名称: (S)-6-amino-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((S)-2-((R)-2-amino-5-guanidinopentanamido)-3-(4-hydroxy-2,6-dimethylphenyl)propanamido)hexanamide
别名: SS-31;MTP-131;Bendavia
SMILES: NC(C(NC(C(NC(C(NC(C(N)=O)CC1C=CC=CC=1)=O)CCCCN)=O)CC1C(C)=CC(O)=CC=1C)=O)CCCNC(=N)N
分子式: C34H60F3N9O7
分子量: 753.81
纯度:
保存条件: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description:
In Vivo:
In Vitro:
References: Elamipretide (SS-31, MTP-131, Bendavia) is a novel cell-permeable antioxidant tetrapeptide (D-Arg-dimethylTyr-Lys-Phe-NH2) that targets inner mitochondrial membrane and prevents oxidative damage of neuronal cells and other cell types; prevents mitochondrial depolarization, reduces islet cell apoptosis, increases islet cell yield, and improves posttransplantation function. Other Indication Phase 3 Clinical
Kinase Assay:
Cell Assay:
Animal Administration:
References:
MSDS
TITLE DOWNLOAD
MSDS_1093_DC21695_736992-21-5
COA
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