Lasmiditan (COL-144; LY573144)
产品编号: DC7710
我们的合作伙伴:
中国地区超过5000个高品质化合物库存
应用领域
Lasmiditan (COL-144; LY573144) is a high-affinity, highly selective 5-HT1F receptor agonist(Ki=2.1 nM), compared with Ki of 1043 nM and 1357 nM at the 5-HT(1B) and 5-HT(1D) receptors, respectively.
Cas No.: |
439239-90-4 |
名称: |
|
别名: |
COL-144; LY-573144,COL144; LY 573144 |
SMILES: |
FC1=CC(F)=C(C(NC2=CC=CC(C(C3CCN(C)CC3)=O)=N2)=O)C(F)=C1 |
分子式: |
C19H18F3N3O2 |
分子量: |
377.36 |
纯度: |
|
保存条件: |
2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
Description: |
|
In Vivo: |
|
In Vitro: |
|
References: |
Lasmiditan (COL-144; LY573144) is a high-affinity, highly selective 5-HT1F receptor agonist(Ki=2.1 nM), compared with Ki of 1043 nM and 1357 nM at the 5-HT(1B) and 5-HT(1D) receptors, respectively.
IC50 value: 2.1 nM (Ki, 5-HT1F); >1000 nM (Ki, 5-HT1B/5- |
Kinase Assay: |
|
Cell Assay: |
|
Animal Administration: |
|
References: |
|
MSDS
TITLE |
DOWNLOAD |
MSDS_3451_DC7710_439239-90-4 |
|
COA
LOT NO. |
DOWNLOAD |
|
|
询盘