SBI993

产品编号: DC11283 Featured
SBI993
结构式
2073059-56-8
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中国地区超过5000个高品质化合物库存
应用领域
SBI-993是SBI-477的类似物,其显示出改善的效力和适合体内生物利用度的药代动力学性质
Cas No.: 2073059-56-8
名称: N-(4-(4-methoxyphenyl)thiazol-2-yl)-4-(2-morpholino-2-oxoethoxy)benzamide
别名: SBI-993,SBI 993,SBI993
SMILES: C(NC1=NC(C2=CC=C(OC)C=C2)=CS1)(=O)C1=CC=C(OCC(N2CCOCC2)=O)C=C1
分子式: C23H23N3O5S
分子量: 453.51
纯度:
保存条件: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description:
In Vivo:
In Vitro:
References: SBI-993 is an analog of SBI-477 that shows improved potency and suitable pharmacokinetic properties for in vivo bioavailability; reduces Txnip and Arrdc4 expression to a degree similar to that seen with SBI-477 in human myotubes; reduces muscle and liver TAG levels, enhances insulin signaling, and improved glucose tolerance in mice fed a high-fat diet.
Kinase Assay:
Cell Assay:
Animal Administration:
References:
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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