XMU-MP-1
产品编号: DC9926
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应用领域
XMU-MP-1是可逆和选择性的 MST1/2 抑制剂，IC50 分别为71.1和38.1 nM。
| Cas No.: |
2061980-01-4 |
| 名称: |
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| 别名: |
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| SMILES: |
CN1C2=C(C(=O)N(C3=CN=C(N=C31)NC4=CC=C(C=C4)S(=O)(=O)N)C)SC=C2 |
| 分子式: |
C17H16N6O3S2 |
| 分子量: |
416.48 |
| 纯度: |
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| 保存条件: |
2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
| Description: |
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| In Vitro: |
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| References: |
XMU-MP-1 is a reversible and selective MST1/2 inhibitor with IC50 values of 71.1 ± 12.9 nM and 38.1 ± 6.9 nM against MST1 and MST2, respectively. XMU-MP-1 also reduces the phosphorylation of LATS1/2, and YAP by inhibiting MST1/2 kinase activities.
In vitr |
| Kinase Assay: |
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| Animal Administration: |
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| References: |
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MSDS
COA
| LOT NO. |
DOWNLOAD |
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| 2018-0101 |
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