DC12654 |
PLX8394
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PLX8394 是一种有效的,选择性的 BRaf 抑制剂,抑制 BRAFV600E 活性的 IC50 值约为 5 nM。 |
DC9743 |
CB1954(Tretazicar)
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CB1954(Tretazicar) in stock,price: 350 USD/100mg. CB1954(Tretazicar) is a anticancer prodrug that is converted in the presence of the enzyme NQO2 and co-substrate caricotamide ( EP-0152R) (EP) into a potent cytotoxic bifunctional alkylating agent.It can |
DC26175 |
NLX-101(F-15599)
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NLX-101(F-15599) is a novel compound that activates serotonin 5-HT1A receptors with exceptional selectivity, having over 1000-fold higher affinity for this target over other receptors. |
DC26173 |
YM-53601
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YM-53601 is a squalene synthase inhibitor (IC50s = 79 and 90 nM in HepG2 cells and rat liver microsomes, respectively). |
DC26160 |
Ethosalamide
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Etosalamide, also known as Ethosalamide, is an antipyretic and analgesics agent. |
DC26155 |
Sulfaphenazole
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Sulfaphenazole is an inhibitor of CYP2C9 (Ki = 0.3 μM) that demonstrates at least 100-fold selectivity over other CYP450 isoforms (Kis = 63 and 29 μM for CYP2C8 and CYP2C18, respectively, and no activity at CYP1A1, CYP1A2, CYP3A4, CYP2C19). |
DC26151 |
Naloxone (hydrochloride)
|
Naloxone is an opioid inverse agonist drug used to counter the effects of opiate overdose. |
DC26139 |
2-(5-Chloro-1H-indol-2-yl)acetic acid
|
2-(5-Chloro-1H-indol-2-yl)acetic acid|CAS 720000-48-6 |
DC12542 |
GOT1 inhibitor 2c
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GOT1抑制剂2c是谷氨酸草酰乙酸转氨酶1(GOT1)的一流的非共价抑制剂,IC50为8.2μM。 |
DC12541 |
iGOT1-01
|
iGOT1-01 is a small molecule inhibitor of aspartate aminotransferase 1 (glutamate oxaloacetate transaminase 1 (GOT1)) with IC50 of 11.3 uM. |