PAK4-IN-1（KPT9274）
产品编号: DC8717
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应用领域
KPT-9274是有口服活性的 PAK4/烟酰胺磷酸核糖基转移酶 (Nampt) 抑制剂，IC50 值分别为小于 100 和 125 nM。
| Cas No.: |
1643913-93-2 |
| 名称: |
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| 别名: |
KPT 9274，KPT9274，KPT-9274 |
| SMILES: |
C1CN(CCC1(F)F)C(=O)C2=CC=C(C=C2)C3=CC(=C4C(=C3)C=C(O4)CNC(=O)/C=C/C5=CN=C(C=C5)N)C6=CC=C(C=C6)F |
| 分子式: |
C35H29F3N4O3 |
| 分子量: |
610.63 |
| 纯度: |
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| 保存条件: |
2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
| Description: |
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| In Vivo: |
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| In Vitro: |
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| References: |
PAK4-IN-1 is an inhibitor of p21-activated kinases (PAKs), with IC50 of ≤100 nM in MTT assay.The detailed information please refer to WO2015003166A1. |
| Kinase Assay: |
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| Cell Assay: |
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| Animal Administration: |
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| References: |
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MSDS
COA
| LOT NO. |
DOWNLOAD |
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| 2018-0101 |
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