YK-11

产品编号: DC10809 Featured
YK-11
结构式
1370003-76-1
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中国地区超过5000个高品质化合物库存
应用领域
YK11 是 androgen 受体的部分激动剂,具有成骨活性。
Cas No.: 1370003-76-1
名称: (17-alpha,20E) 17,20-[(1-methoxyethylidene)bis(oxy)] 3-oxo-19-norpregna-4,20-diene 21-carboxylic acid methyl ester
别名: YK11,YK 11
SMILES: C[C@]12CC[C@H]3[C@H]([C@@H]1CC[C@]24/C(=C\C(=O)OC)/OC(O4)(C)OC)CCC5=CC(=O)CC[C@H]35
分子式: C25H34O6
分子量: 430.53
纯度:
保存条件: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description:
In Vivo:
In Vitro:
References: YK11, known as YK-11, or (17-alpha,20E) 17,20-[(1-methoxyethylidene)bis(oxy)] 3-oxo-19-norpregna-4,20-diene 21-carboxylic acid methyl ester as its chemical name, is the newest ingredient in the SARMs family in recent years. YK11 is said to be the most potent SARM without serious side effects such as hair loss, aggression, prostate enlargement, etc. DHT is something people talk with when come across YK11. YK-11 is derivative from the steroid DHT, so that as partial agonist from the androgen receptor it might activate the androgen receptor to provide a submaximal response when insufficient levels of DHT or Test can be found. In the existence of overstimulation of androgen receptors say when excess levels of DHT or Test can be found YK-11 will behave as an aggressive inhibitor of androgen receptors . It is because partial agonists typically display both agonistic and hostile properties.YK11 is claimed to be the most powerful among all SARMs, much more potent than classic anabolic steroids like DHT. YK11 is thought to be a SARM and generate the result of myostatin simultaneously. YK11 is much more anabolic and androgenic when in comparison to a different popular solution, DHTwhich is really a steroid di-hydrotestosterone with some adverse effects. These negative effects are mentioned above, including hair loss as well as prostate enlargement.however, with YK11 you do not have any of these problems. Actually, some research has proven that YK11 can really enable you to grow more hair and also the prostate hasn’t altered whatsoever in the trials carried out in the experiments.Myostatin is a protein that, when it is within the body, myostatin restricts the muscle tissue growth and production. In this way, myostatin is bad to bodybuilders. By inhibiting myostatin, YK11 induces muscle cells to make more follistatin, and bodybuilders can experience significantly more muscle mass and exponential strength increases. In this sense, YK11 can be as good as testosterone in terms of muscle strengthening.In addition, YK-11 is an androgen. YK11 attaches itself to the AR (androgen receptor), and has been discovered that muscle cells produce more anabolic factors if exposed to 500 nmol (nanomoles) YK11 than if you expose the same muscle cells to 500 nmol DHT. YK11 fortifies parts of your muscles in the same manner as testosterone and the only difference isthat it doesn’t have the additional side-effect. The primary factor to keep in mind about YK11 is it may also provide you with a strengthening boost when you’re during a workout session so apply for longer without encountering any fatigue. On the top of that, it may also help you to modify your body genetics so that you can build more muscle and faster than before.
Kinase Assay:
Cell Assay:
Animal Administration:
References:
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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