Cas No.: | 1260907-17-2 |
名称: | (S)-2-(6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-4-yl)-N-ethylacetamide |
别名: | I-BET-762,GSK525762,GSK-525762,GSK 525762 |
SMILES: | N12C(C)=NN=C1[C@@H](CC(NCC)=O)N=C(C1=CC=C(Cl)C=C1)C1=CC(OC)=CC=C12 |
分子式: | C22H22ClN5O2 |
分子量: | 423.9 |
纯度: | |
保存条件: | 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
Description: | |
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References: | GSK525762 is a small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family of bromodomain-containing proteins with potential antineoplastic activity. Upon administration, the BET inhibitor GSK525762 binds to the acetylated lysine recogniti |
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