MG-101
产品编号: DC7702
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应用领域
MG-101是有效的半胱氨酸蛋白酶抑制剂，抑制钙蛋白酶I，钙蛋白酶II，组织蛋白酶B和组织蛋白酶L的Ki分别为190，220，150和500 pM。
| Cas No.: |
110044-82-1 |
| 名称: |
N-Acetyl-L-leucine-L-leucine-L-norleucinal |
| 别名: |
Calpain inhibitor-1,MG101，MG-101，MG 101 |
| SMILES: |
O=C(N[C@H](C=O)CCCC)[C@@H](NC([C@@H](NC(C)=O)CC(C)C)=O)CC(C)C |
| 分子式: |
C20H37N3O4 |
| 分子量: |
383.53 |
| 纯度: |
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| 保存条件: |
2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
| Description: |
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| In Vitro: |
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| References: |
Calpain inhibitor (IC50 = 0.09 μM) that activates p53-dependent apoptosis in tumor cell lines. Increases activated p53, p21 and caspase levels and promotes cell cycle arrest through inhibition of cyclin D degradation in vitro. Also attenuates ischemia/rep |
| Kinase Assay: |
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| Cell Assay: |
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| Animal Administration: |
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| References: |
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MSDS
| TITLE |
DOWNLOAD |
| MSDS_1912_DC7702_110044-82-1 |
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COA
| LOT NO. |
DOWNLOAD |
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询盘
