LYS6K2(LY2584702) tosylate salt
产品编号: DC7943
Featured
我们的合作伙伴:
中国地区超过5000个高品质化合物库存
应用领域
LY-2584702 tosylate salt 是一种 ATP 竞争性的选择性 p70S6K 抑制剂，IC50 为 4 nM。LY-2584702 抑制 S6K1 的 IC50 为 2 nM。
| Cas No.: |
1082949-68-5 |
| 名称: |
4-[4-[4-[4-fluoro-3-(trifluoromethyl)phenyl]-1-methyl-imidazol-2-yl]-1-piperidyl]-1H-pyrazolo[3,4-d]pyrimidine |
| 别名: |
LY-2584702，LY 2584702,LYS6K2 |
| SMILES: |
C1=NC(N2CCC(C3N(C)C=C(C4=CC=C(F)C(C(F)(F)F)=C4)N=3)CC2)=C2C=NNC2=N1.C(S(O)(=O)=O)1=CC=C(C)C=C1 |
| 分子式: |
C28H27F4N7O3S |
| 分子量: |
617.62 |
| 纯度: |
|
| 保存条件: |
2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
| Description: |
|
| In Vivo: |
|
| In Vitro: |
|
| References: |
LY-2584702 is an orally available inhibitor of p70S6K signaling, with potential antineoplastic activity. LY2584702 inhibits ribosomal protein S6 Kinase (p70S6K), and prevents phosphorylation of the S6 subunit of ribosomes, thereby inhibiting normal riboso |
| Kinase Assay: |
|
| Cell Assay: |
|
| Animal Administration: |
|
| References: |
|
MSDS
COA
| LOT NO. |
DOWNLOAD |
|
|
| 2018-0101 |
|
询盘
