2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
生物活性
Description
In Vivo
In Vitro
化合物的使用
Kinase Assay
Cell Assay
Animal Administration
参考文献
MPEP is a potent and highly selective non-competitive antagonist at the mGlu5 receptor subtype (IC50 = 36 nM) and a positive allosteric modulator at mGlu4 receptors. Centrally active following systemic administration in vivo. Reverses mechanical hyperalgesia in the inflamed rat hind paw. For the detailed information about the solubility of MPEP in water, the solubility of MPEP in DMSO, the solubility of MPEP in PBS buffer, the animal experiment（test） of MPEP,the in vivo,in vitro and clinical trial test of MPEP,the cell experiment（test） of MPEP,the IC50, EC50 and Affinity of MPEP, please contact DC Chemicals.
